Abstract

Enzyme inhibition plays a central role in drug discovery and development, offering a powerful strategy for modulating biological pathways and treating a wide range of diseases. This article provides an overview of enzyme inhibition, elucidating the molecular mechanisms involved, exploring the diverse applications in medicine and biotechnology, and highlighting the therapeutic implications for various disorders. From small molecule inhibitors to biologics and beyond, understanding the principles of enzyme inhibition is essential for the rational design of effective therapeutics.